Noab BioDiscoveries - Shaping Drug Discovery

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October 2003; 31 (10)   [Index by Author]  [Cover Caption]
       Articles
       Short Communications
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Articles:

L.-J. Chen, E. H. Lebetkin, and L. T. Burka
METABOLISM OF (R)-(+)-MENTHOFURAN IN FISCHER-344 RATS: IDENTIFICATION OF SULFONIC ACID METABOLITES
Drug Metab Dispos 2003 31: 1208-1213. [Abstract] [Full Text] [PDF]  

Debbie Tam, Huadong Sun, and K. Sandy Pang
INFLUENCE OF P-GLYCOPROTEIN, TRANSFER CLEARANCES, AND DRUG BINDING ON INTESTINAL METABOLISM IN CACO-2 CELL MONOLAYERS OR MEMBRANE PREPARATIONS: A THEORETICAL ANALYSIS
Drug Metab Dispos 2003 31: 1214-1226. [Abstract] [Full Text] [PDF]  

Kyoung-Ah Kim, Min-Jung Kim, Ji-Young Park, Ji-Hong Shon, Young-Ran Yoon, Sang-Seop Lee, Kwang-Hyeon Liu, Jin-Ho Chun, Myung-Ho Hyun, and Jae-Gook Shin
STEREOSELECTIVE METABOLISM OF LANSOPRAZOLE BY HUMAN LIVER CYTOCHROME P450 ENZYMES
Drug Metab Dispos 2003 31: 1227-1234. [Abstract] [Full Text] [PDF]  

Kohji Takara, Noriaki Ohnishi, Sayo Horibe, and Teruyoshi Yokoyama
EXPRESSION PROFILES OF DRUG-METABOLIZING ENZYME CYP3A AND DRUG EFFLUX TRANSPORTER MULTIDRUG RESISTANCE 1 SUBFAMILY mRNAS IN RAT SMALL INTESTINE
Drug Metab Dispos 2003 31: 1235-1239. [Abstract] [Full Text] [PDF]  

Amit S. Kalgutkar, Hang T. Nguyen, Alfin D. N. Vaz, Anke Doan, Deepak K. Dalvie, Dale G. McLeod, and John C. Murray
IN VITRO METABOLISM STUDIES ON THE ISOXAZOLE RING SCISSION IN THE ANTI-INFLAMMATORY AGENT LEFLUNOMIDE TO ITS ACTIVE {alpha}-CYANOENOL METABOLITE A771726: MECHANISTIC SIMILARITIES WITH THE CYTOCHROME P450-CATALYZED DEHYDRATION OF ALDOXIMES
Drug Metab Dispos 2003 31: 1240-1250. [Abstract] [Full Text] [PDF]  

Tomoyuki Ohe, Masahiko Sato, Sachiko Tanaka, Naoko Fujino, Mikiko Hata, Yoshihiro Shibata, Akio Kanatani, Takehiro Fukami, Masayo Yamazaki, Masato Chiba, and Yasuyuki Ishii
EFFECT OF P-GLYCOPROTEIN-MEDIATED EFFLUX ON CEREBROSPINAL FLUID/PLASMA CONCENTRATION RATIO
Drug Metab Dispos 2003 31: 1251-1254. [Abstract] [Full Text] [PDF]  

Bang-Ning Yu, Guo-Lin Chen, Nan He, Dong-Sheng Ouyang, Xiao-Ping Chen, Zhao-Qian Liu, and Hong-Hao Zhou
PHARMACOKINETICS OF CITALOPRAM IN RELATION TO GENETIC POLYMORPHISM OF CYP2C19
Drug Metab Dispos 2003 31: 1255-1259. [Abstract] [Full Text] [PDF]  

Sang K. Kim, Kimberley J. Woodcroft, Sang G. Kim, and Raymond F. Novak
INSULIN AND GLUCAGON SIGNALING IN REGULATION OF MICROSOMAL EPOXIDE HYDROLASE EXPRESSION IN PRIMARY CULTURED RAT HEPATOCYTES
Drug Metab Dispos 2003 31: 1260-1268. [Abstract] [Full Text] [PDF]  

Maria G. Beconi, Ann Mao, David Q. Liu, Christopher Kochansky, Tony Pereira, Conrad Raab, Paul Pearson, and Shuet-Hing Lee Chiu
METABOLISM AND PHARMACOKINETICS OF A DIPEPTIDYL PEPTIDASE IV INHIBITOR IN RATS, DOGS, AND MONKEYS WITH SELECTIVE CARBAMOYL GLUCURONIDATION OF THE PRIMARY AMINE IN DOGS
Drug Metab Dispos 2003 31: 1269-1277. [Abstract] [Full Text] [PDF]  

Short Communications:

John R. Jalas, Xinxin Ding, and Sharon E. Murphy
COMPARATIVE METABOLISM OF THE TOBACCO-SPECIFIC NITROSAMINES 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE AND 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANOL BY RAT CYTOCHROME P450 2A3 AND HUMAN CYTOCHROME P450 2A13
Drug Metab Dispos 2003 31: 1199-1202. [Abstract] [Full Text] [PDF]  

Michael H. Lumpkin, James V. Bruckner, Jerry L. Campbell, Cham E. Dallas, Catherine A. White, and Jeffrey W. Fisher
PLASMA BINDING OF TRICHLOROACETIC ACID IN MICE, RATS, AND HUMANS UNDER CANCER BIOASSAY AND ENVIRONMENTAL EXPOSURE CONDITIONS
Drug Metab Dispos 2003 31: 1203-1207. [Abstract] [Full Text] [PDF]  

To see an article, click its [Full Text] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.


Cover Caption:

Expression profiles for CYP3A and mdr1 subfamily mRNAs in rat liver (A) and small intestine (B) by RT-PCR. See the article by Takara et al. on page 1235 of this issue.



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