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Other Issues:
September 2003; 31 (9)   [Index by Author]  [Cover Caption]
       Articles
       Commentaries
       Short Communications
       Erratum
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Articles:

Jarmo S. Salonen, Leena Nyman, Alan R. Boobis, Robert J. Edwards, Patricia Watts, Brian G. Lake, Roger J. Price, Anthony B. Renwick, Maria-José Gómez-Lechón, José V. Castell, Magnus Ingelman-Sundberg, Mats Hidestrand, Andre Guillouzo, Laurent Corcos, Peter S. Goldfarb, David F.V. Lewis, Päivi Taavitsainen, and Olavi Pelkonen
COMPARATIVE STUDIES ON THE CYTOCHROME P450-ASSOCIATED METABOLISM AND INTERACTION POTENTIAL OF SELEGILINE BETWEEN HUMAN LIVER-DERIVED IN VITRO SYSTEMS
Drug Metab Dispos 2003 31: 1093-1102. [Abstract] [Full Text] [PDF]  

Lisa A. McConnachie, Brian Phillips, Manoj Bajpai, Danny D. Shen, and Rodney J. Y. Ho
ONLY TRUNCATED, NOT COMPLETE CYTOCHROME P450 2D6 RNA TRANSCRIPT AND NO DETECTABLE ENZYME ACTIVITY ARE EXPRESSED IN HUMAN LYMPHOCYTES
Drug Metab Dispos 2003 31: 1103-1107. [Abstract] [Full Text] [PDF]  

Aleksandra Galetin, Stephen E. Clarke, and J. Brian Houston
MULTISITE KINETIC ANALYSIS OF INTERACTIONS BETWEEN PROTOTYPICAL CYP3A4 SUBGROUP SUBSTRATES: MIDAZOLAM, TESTOSTERONE, AND NIFEDIPINE
Drug Metab Dispos 2003 31: 1108-1116. [Abstract] [Full Text] [PDF]  

Tiia Kuuranne, Mika Kurkela, Mario Thevis, Wilhelm Schänzer, Moshe Finel, and Risto Kostiainen
GLUCURONIDATION OF ANABOLIC ANDROGENIC STEROIDS BY RECOMBINANT HUMAN UDP-GLUCURONOSYLTRANSFERASES
Drug Metab Dispos 2003 31: 1117-1124. [Abstract] [Full Text] [PDF]  

Michael H. Court, Soundarajan Krishnaswamy, Qin Hao, Su X. Duan, Christopher J. Patten, Lisa L. von Moltke, and David J. Greenblatt
EVALUATION OF 3'-AZIDO-3'-DEOXYTHYMIDINE, MORPHINE, AND CODEINE AS PROBE SUBSTRATES FOR UDP-GLUCURONOSYLTRANSFERASE 2B7 (UGT2B7) IN HUMAN LIVER MICROSOMES: SPECIFICITY AND INFLUENCE OF THE UGT2B7*2 POLYMORPHISM
Drug Metab Dispos 2003 31: 1125-1133. [Abstract] [Full Text] [PDF]  

Graeme B. J. Smith, John R. Bend, Leanne L. Bedard, Ken R. Reid, Dimitri Petsikas, and Thomas E. Massey
BIOTRANSFORMATION OF 4-(METHYLNITROSAMINO)-1-(3-PYRIDYL)-1-BUTANONE (NNK) IN PERIPHERAL HUMAN LUNG MICROSOMES
Drug Metab Dispos 2003 31: 1134-1141. [Abstract] [Full Text] [PDF]  

R. J. Lantz, T. A. Gillespie, T. J. Rash, F. Kuo, M. Skinner, H-Y. Kuan, and M. P. Knadler
METABOLISM, EXCRETION, AND PHARMACOKINETICS OF DULOXETINE IN HEALTHY HUMAN SUBJECTS
Drug Metab Dispos 2003 31: 1142-1150. [Abstract] [Full Text] [PDF]  

Brendan M. Johnson, William N. Charman, and Christopher J. H. Porter
APPLICATION OF COMPARTMENTAL MODELING TO AN EXAMINATION OF IN VITRO INTESTINAL PERMEABILITY DATA: ASSESSING THE IMPACT OF TISSUE UPTAKE, P-GLYCOPROTEIN, AND CYP3A
Drug Metab Dispos 2003 31: 1151-1160. [Abstract] [Full Text] [PDF]  

Magang Shou, Ryan Norcross, Grit Sandig, Ping Lu, Yinghe Li, Yuh Lin, Qin Mei, A. David Rodrigues, and Thomas H. Rushmore
SUBSTRATE SPECIFICITY AND KINETIC PROPERTIES OF SEVEN HETEROLOGOUSLY EXPRESSED DOG CYTOCHROMES P450
Drug Metab Dispos 2003 31: 1161-1169. [Abstract] [Full Text] [PDF]  

Gang Luo, Jianrong Lin, William D. Fiske, Renke Dai, Tian J. Yang, Sean Kim, Michael Sinz, Edward LeCluyse, Eric Solon, James M. Brennan, Irma H. Benedek, Summer Jolley, Darryl Gilbert, Lifei Wang, Frank W. Lee, and Liang-Shang Gan
CONCURRENT INDUCTION AND MECHANISM-BASED INACTIVATION OF CYP3A4 BY AN L-VALINAMIDE DERIVATIVE
Drug Metab Dispos 2003 31: 1170-1175. [Abstract] [Full Text] [PDF]  

A. L. Slitt, N. J. Cherrington, J. M. Maher, and C. D. Klaassen
INDUCTION OF MULTIDRUG RESISTANCE PROTEIN 3 IN RAT LIVER IS ASSOCIATED WITH ALTERED VECTORIAL EXCRETION OF ACETAMINOPHEN METABOLITES
Drug Metab Dispos 2003 31: 1176-1186. [Abstract] [Full Text] [PDF]  

Jyrki Taskinen, Brian T. Ethell, Pia Pihlavisto, Alan M. Hood, Brian Burchell, and Michael W. H. Coughtrie
CONJUGATION OF CATECHOLS BY RECOMBINANT HUMAN SULFOTRANSFERASES, UDP-GLUCURONOSYLTRANSFERASES, AND SOLUBLE CATECHOL O-METHYLTRANSFERASE: STRUCTURE-CONJUGATION RELATIONSHIPS AND PREDICTIVE MODELS
Drug Metab Dispos 2003 31: 1187-1197. [Abstract] [Full Text] [PDF]  

Commentaries:

Ronald N. Hines
PUBLICATION OF STAND-ALONE SINGLE NUCLEOTIDE POLYMORPHISM (SNP) DISCOVERY DATA
Drug Metab Dispos 2003 31: 1073. [Full Text] [PDF]  

Short Communications:

Meena R. Sharma, Parameswaran Periandythevar, and Bernard H. Shapiro
SPURIOUS OBSERVATION OF SPLENIC CYP2B1 EXPRESSION
Drug Metab Dispos 2003 31: 1074-1076. [Abstract] [Full Text] [PDF]  

Sean Ekins, Jennifer Berbaum, and Richard K. Harrison
GENERATION AND VALIDATION OF RAPID COMPUTATIONAL FILTERS FOR CYP2D6 AND CYP3A4
Drug Metab Dispos 2003 31: 1077-1080. [Abstract] [Full Text] [PDF]  

Xiuling Zhang, Ying Chen, Yiqin Liu, Xiang Ren, Qing-Yu Zhang, Michele Caggana, and Xinxin Ding
SINGLE NUCLEOTIDE POLYMORPHISMS OF THE HUMAN CYP2A13 GENE: EVIDENCE FOR A NULL ALLELE
Drug Metab Dispos 2003 31: 1081-1085. [Abstract] [Full Text] [PDF]  

Andrew N. Stone, Peter I. Mackenzie, Aleksandra Galetin, J. Brian Houston, and John O. Miners
ISOFORM SELECTIVITY AND KINETICS OF MORPHINE 3- AND 6-GLUCURONIDATION BY HUMAN UDP-GLUCURONOSYLTRANSFERASES: EVIDENCE FOR ATYPICAL GLUCURONIDATION KINETICS BY UGT2B7
Drug Metab Dispos 2003 31: 1086-1089. [Abstract] [Full Text] [PDF]  

Kyoung-Ah Kim and Ji-Young Park
INHIBITORY EFFECT OF GLYBURIDE ON HUMAN CYTOCHROME P450 ISOFORMS IN HUMAN LIVER MICROSOMES
Drug Metab Dispos 2003 31: 1090-1092. [Abstract] [Full Text] [PDF]  

Erratum:

CORRECTION TO "DETECTION OF CARBOXYLIC ACIDS AND INHIBITION OF HIPPURIC ACID FORMATION IN RATS TREATED WITH 3-BUTENE-1,2-DIOL, A MAJOR METABOLITE OF 1,3-BUTADIENE"
Drug Metab Dispos 2003 31: 1198. [Full Text] [PDF]  

To see an article, click its [Full Text] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.


Cover Caption:

Immunohistochemical detection of Mrp3 in liver following PB, DAS, OLT, or TSO administration. See the article by Slitt et al. on page 1176 of this issue.



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