DMD Noab BioDiscoveries - Shaping Drug Discovery

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July 2004; 32 (7)   [Index by Author]  [Cover Caption]
       Articles
       Short Communications
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Articles:

Hai-Zhi Bu, William F. Pool, Ellen Y. Wu, Susan R. Raber, Michael A. Amantea, and Bhasker V. Shetty
METABOLISM AND EXCRETION OF CAPRAVIRINE, A NEW NON-NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITOR, ALONE AND IN COMBINATION WITH RITONAVIR IN HEALTHY VOLUNTEERS
Drug Metab Dispos 2004 32: 689-698. [Abstract] [Full Text] [PDF]  

M. Teresa Donato, Nuria Jiménez, José V. Castell, and M. José Gómez-Lechón
FLUORESCENCE-BASED ASSAYS FOR SCREENING NINE CYTOCHROME P450 (P450) ACTIVITIES IN INTACT CELLS EXPRESSING INDIVIDUAL HUMAN P450 ENZYMES
Drug Metab Dispos 2004 32: 699-706. [Abstract] [Full Text] [PDF]  

Takashi Ashino, Takiko Oguro, Seiji Shioda, Reiko Horai, Masahide Asano, Kenji Sekikawa, Yoichiro Iwakura, Satoshi Numazawa, and Takemi Yoshida
INVOLVEMENT OF INTERLEUKIN-6 AND TUMOR NECROSIS FACTOR {alpha} IN CYP3A11 AND 2C29 DOWN-REGULATION BY BACILLUS CALMETTE-GUÉRIN AND LIPOPOLYSACCHARIDE IN MOUSE LIVER
Drug Metab Dispos 2004 32: 707-714. [Abstract] [Full Text] [PDF]  

Tommy B. Andersson, Eva Bredberg, Hans Ericsson, and Helena Sjöberg
AN EVALUATION OF THE IN VITRO METABOLISM DATA FOR PREDICTING THE CLEARANCE AND DRUG-DRUG INTERACTION POTENTIAL OF CYP2C9 SUBSTRATES
Drug Metab Dispos 2004 32: 715-721. [Abstract] [Full Text] [PDF]  

Joseph W. Polli, Todd M. Baughman, Joan E. Humphreys, Kelly H. Jordan, Angela L. Mote, Lindsey O. Webster, Robert J. Barnaby, Giovanni Vitulli, Luigina Bertolotti, Kevin D. Read, and Cosette J. Serabjit-Singh
THE SYSTEMIC EXPOSURE OF AN N-METHYL-D-ASPARTATE RECEPTOR ANTAGONIST IS LIMITED IN MICE BY THE P-GLYCOPROTEIN AND BREAST CANCER RESISTANCE PROTEIN EFFLUX TRANSPORTERS
Drug Metab Dispos 2004 32: 722-726. [Abstract] [Full Text] [PDF]  

Samuel M. Poloyac, Michael A. Tortorici, Danielle I. Przychodzin, Robert B. Reynolds, Wen Xie, Reginald F. Frye, and Michael A. Zemaitis
THE EFFECT OF ISONIAZID ON CYP2E1- AND CYP4A-MEDIATED HYDROXYLATION OF ARACHIDONIC ACID IN THE RAT LIVER AND KIDNEY
Drug Metab Dispos 2004 32: 727-733. [Abstract] [Full Text] [PDF]  

Nathan J. Cherrington, Angela L. Slitt, Ning Li, and Curtis D. Klaassen
LIPOPOLYSACCHARIDE-MEDIATED REGULATION OF HEPATIC TRANSPORTER mRNA LEVELS IN RATS
Drug Metab Dispos 2004 32: 734-741. [Abstract] [Full Text] [PDF]  

Eszter Hazai, Peter V. Gagne, and David Kupfer
GLUCURONIDATION OF THE OXIDATIVE CYTOCHROME P450-MEDIATED PHENOLIC METABOLITES OF THE ENDOCRINE DISRUPTOR PESTICIDE: METHOXYCHLOR BY HUMAN HEPATIC UDP-GLUCURONOSYL TRANSFERASES
Drug Metab Dispos 2004 32: 742-751. [Abstract] [Full Text] [PDF] Correction  

Ying Zhang, Teruaki Akao, Norio Nakamura, Masao Hattori, Xiu-Wei Yang, Chang-Ling Duan, and Jian-Xun Liu
MAGNESIUM LITHOSPERMATE B IS EXCRETED RAPIDLY INTO RAT BILE MOSTLY AS METHYLATED METABOLITES, WHICH ARE POTENT ANTIOXIDANTS
Drug Metab Dispos 2004 32: 752-757. [Abstract] [Full Text] [PDF]  

Junichi Narukawa, Hiroki Inoue, Seiyu Kato, and Hiroshi Yokota
GLUCURONIDATION OF 1-NAPHTHOL AND EXCRETION INTO THE VEIN IN PERFUSED RAT KIDNEY
Drug Metab Dispos 2004 32: 758-761. [Abstract] [Full Text] [PDF]  

Toshiki Tabata, Miki Katoh, Shogo Tokudome, Masakiyo Hosakawa, Kan Chiba, Miki Nakajima, and Tsuyoshi Yokoi
BIOACTIVATION OF CAPECITABINE IN HUMAN LIVER: INVOLVEMENT OF THE CYTOSOLIC ENZYME ON 5'-DEOXY-5-FLUOROCYTIDINE FORMATION
Drug Metab Dispos 2004 32: 762-767. [Abstract] [Full Text] [PDF]  

Nikhil K. Basu, Labanyamoy Kole, Shigeki Kubota, and Ida S. Owens
HUMAN UDP-GLUCURONOSYLTRANSFERASES SHOW ATYPICAL METABOLISM OF MYCOPHENOLIC ACID AND INHIBITION BY CURCUMIN
Drug Metab Dispos 2004 32: 768-773. [Abstract] [Full Text] [PDF]  

Short Communications:

Kristina K. Wolf, Sheryl G. Wood, Jenna L. Bement, Peter R. Sinclair, Steven A. Wrighton, Elizabeth Jeffery, Frank J. Gonzalez, and Jacqueline F. Sinclair
ROLE OF MOUSE CYP2E1 IN THE O-HYDROXYLATION OF P-NITROPHENOL: COMPARISON OF ACTIVITIES IN HEPATIC MICROSOMES FROM CYP2E1(-/-) AND WILD-TYPE MICE
Drug Metab Dispos 2004 32: 681-684. [Abstract] [Full Text] [PDF]  

Yoko Yasunami, Hirokazu Hara, Tatsunori Iwamura, Tadashi Kataoka, and Tetsuo Adachi
C-JUN N-TERMINAL KINASE MODULATES 1,25-DIHYDROXYVITAMIN D3-INDUCED CYTOCHROME P450 3A4 GENE EXPRESSION
Drug Metab Dispos 2004 32: 685-688. [Abstract] [Full Text] [PDF]  

To see an article, click its [Full Text] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.


Cover Caption:

Proposed metabolic pathway of capecitabine in humans. See the article by Tabata et al. on page 742 of this issue.



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