DMD Celsis microsomes mean better data

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February 2005; 33 (2)   [Index by Author]  [Cover Caption]
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Articles:

Christian Zimmermann, Heike Gutmann, Petr Hruz, Jean-Pierre Gutzwiller, Christoph Beglinger, and Juergen Drewe
MAPPING OF MULTIDRUG RESISTANCE GENE 1 AND MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN ISOFORM 1 TO 5 mRNA EXPRESSION ALONG THE HUMAN INTESTINAL TRACT
Drug Metab Dispos 2005 33: 219-224. Published online November 2, 2004; 10.1124/dmd.104.001354 [Abstract] [Full Text] [PDF]  

Mizuki Ninomiya, Kousei Ito, and Toshiharu Horie
FUNCTIONAL ANALYSIS OF DOG MULTIDRUG RESISTANCE-ASSOCIATED PROTEIN 2 (MRP2) IN COMPARISON WITH RAT MRP2
Drug Metab Dispos 2005 33: 225-232. Published online October 26, 2004; 10.1124/dmd.104.002196 [Abstract] [Full Text] [PDF]  

Anna Phillips, Steve R. Hood, G. Gordon Gibson, and Nick J. Plant
IMPACT OF TRANSCRIPTION FACTOR PROFILE AND CHROMATIN CONFORMATION ON HUMAN HEPATOCYTE CYP3A GENE EXPRESSION
Drug Metab Dispos 2005 33: 233-242. Published online November 2, 2004; 10.1124/dmd.104.001461 [Abstract] [Full Text] [PDF]  

Amit S. Kalgutkar, Alfin D. N. Vaz, Mary E. Lame, Kirk R. Henne, John Soglia, Sabrina X. Zhao, Yuri A. Abramov, Franco Lombardo, Claire Collin, Zachary S. Hendsch, and Cornelis E. C. A. Hop
BIOACTIVATION OF THE NONTRICYCLIC ANTIDEPRESSANT NEFAZODONE TO A REACTIVE QUINONE-IMINE SPECIES IN HUMAN LIVER MICROSOMES AND RECOMBINANT CYTOCHROME P450 3A4
Drug Metab Dispos 2005 33: 243-253. Published online November 2, 2004; 10.1124/dmd.104.001735 [Abstract] [Full Text] [PDF] Erratum  

Sukhwinder S. Lakhman, Debashis Ghosh, and Javier G. Blanco
FUNCTIONAL SIGNIFICANCE OF A NATURAL ALLELIC VARIANT OF HUMAN CARBONYL REDUCTASE 3 (CBR3)
Drug Metab Dispos 2005 33: 254-257. Published online November 10, 2004; 10.1124/dmd.104.002006 [Abstract] [Full Text] [PDF]  

Ziping Bao, Xiao-Yang He, Xinxin Ding, Saileta Prabhu, and Jun-Yan Hong
METABOLISM OF NICOTINE AND COTININE BY HUMAN CYTOCHROME P450 2A13
Drug Metab Dispos 2005 33: 258-261. Published online November 4, 2004; 10.1124/dmd.104.002105 [Abstract] [Full Text] [PDF]  

R. Scott Obach, Loretta M. Cox, and Larry M. Tremaine
SERTRALINE IS METABOLIZED BY MULTIPLE CYTOCHROME P450 ENZYMES, MONOAMINE OXIDASES, AND GLUCURONYL TRANSFERASES IN HUMAN: AN IN VITRO STUDY
Drug Metab Dispos 2005 33: 262-270. Published online November 16, 2004; 10.1124/dmd.104.002428 [Abstract] [Full Text] [PDF]  

Jane R. Kenny, James L. Maggs, Justice N. A. Tettey, Andrew W. Harrell, Steven G. Parker, Stephen E. Clarke, and B. Kevin Park
FORMATION AND PROTEIN BINDING OF THE ACYL GLUCURONIDE OF A LEUKOTRIENE B4 ANTAGONIST (SB-209247): RELATION TO SPECIES DIFFERENCES IN HEPATOTOXICITY
Drug Metab Dispos 2005 33: 271-281. Published online November 2, 2004; 10.1124/dmd.104.001677 [Abstract] [Full Text] [PDF]  

Robert P. Hanzlik, Stephen C. Fowler, and Janis T. Eells
ABSORPTION AND ELIMINATION OF FORMATE FOLLOWING ORAL ADMINISTRATION OF CALCIUM FORMATE IN FEMALE HUMAN SUBJECTS
Drug Metab Dispos 2005 33: 282-286. Published online November 16, 2004; 10.1124/dmd.104.001289 [Abstract] [Full Text] [PDF]  

Keith A. Hoffmaster, Maciej J. Zamek-Gliszczynski, Gary M. Pollack, and Kim L. R. Brouwer
MULTIPLE TRANSPORT SYSTEMS MEDIATE THE HEPATIC UPTAKE AND BILIARY EXCRETION OF THE METABOLICALLY STABLE OPIOID PEPTIDE [D-PENICILLAMINE2,5]ENKEPHALIN
Drug Metab Dispos 2005 33: 287-293. Published online November 4, 2004; 10.1124/dmd.104.001420 [Abstract] [Full Text] [PDF]  

Short Communications:

Nirmala Raghavan, Donglu Zhang, Mingshe Zhu, Jianing Zeng, and Lisa Christopher
CYP2D6 CATALYZES 5-HYDROXYLATION OF 1-(2-PYRIMIDINYL)-PIPERAZINE, AN ACTIVE METABOLITE OF SEVERAL PSYCHOACTIVE DRUGS, IN HUMAN LIVER MICROSOMES
Drug Metab Dispos 2005 33: 203-208. Published online October 26, 2004; 10.1124/dmd.104.001198 [Abstract] [Full Text] [PDF]  

Kwang-Hyeon Liu, Min-Jung Kim, Woo Moon Jung, Wonku Kang, In-June Cha, and Jae-Gook Shin
LANSOPRAZOLE ENANTIOMER ACTIVATES HUMAN LIVER MICROSOMAL CYP2C9 CATALYTIC ACTIVITY IN A STEREOSPECIFIC AND SUBSTRATE-SPECIFIC MANNER
Drug Metab Dispos 2005 33: 209-213. Published online November 10, 2004; 10.1124/dmd.104.001438 [Abstract] [Full Text] [PDF]  

Bjarte Furnes and Daniel Schlenk
EXTRAHEPATIC METABOLISM OF CARBAMATE AND ORGANOPHOSPHATE THIOETHER COMPOUNDS BY THE FLAVIN-CONTAINING MONOOXYGENASE AND CYTOCHROME P450 SYSTEMS
Drug Metab Dispos 2005 33: 214-218. Published online November 16, 2004; 10.1124/dmd.104.000984 [Abstract] [Full Text] [PDF]  

To see an article, click its [Full Text] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.


Cover Caption:

The three-dimensional structure of porcine testicular carbonyl reductase (PTCR) in green with modeled human CBR3 in yellow, shown at the site of V244M substitution. See the article by Lakhman et al. on page 254 of this issue.



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