DMD Celsis microsomes mean better data

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August 2005; 33 (8)   [Index by Author]  [Cover Caption]
       Symposium Reports
       Articles
       Short Communications
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Symposium Reports:

David S. Riddick, Chunja Lee, Shairoz Ramji, Edwin C. Chinje, Rachel L. Cowen, Kaye J. Williams, Adam V. Patterson, Ian J. Stratford, Charles S. Morrow, Alan J. Townsend, Youssef Jounaidi, Chong-Sheng Chen, Ting Su, Hong Lu, Pamela S. Schwartz, and David J. Waxman
CANCER CHEMOTHERAPY AND DRUG METABOLISM
Drug Metab Dispos 2005 33: 1083-1096. [Abstract] [Full Text] [PDF]  

Articles:

Roger J. Laham, Mark Post, Mehrdad Rezaee, Laurel Donnell-Fink, Joanna J. Wykrzykowska, Seung U. Lee, Donald S. Baim, and Frank W. Sellke
TRANSENDOCARDIAL AND TRANSEPICARDIAL INTRAMYOCARDIAL FIBROBLAST GROWTH FACTOR-2 ADMINISTRATION: MYOCARDIAL AND TISSUE DISTRIBUTION
Drug Metab Dispos 2005 33: 1101-1107. Published online May 6, 2005; 10.1124/dmd.104.002774 [Abstract] [Full Text] [PDF]  

Jürgen Borlak, Maren Blickwede, Tanja Hansen, Wolfgang Koch, Markus Walles, and Karsten Levsen
METABOLISM OF VERAPAMIL IN CULTURES OF RAT ALVEOLAR EPITHELIAL CELLS AND PHARMACOKINETICS AFTER ADMINISTRATION BY INTRAVENOUS AND INHALATION ROUTES
Drug Metab Dispos 2005 33: 1108-1114. Published online May 10, 2005; 10.1124/dmd.105.003723 [Abstract] [Full Text] [PDF]  

Yoichi Kohno, Shigeyuki Kitamura, Seigo Sanoh, Kazumi Sugihara, Nariaki Fujimoto, and Shigeru Ohta
METABOLISM OF THE {alpha},ß-UNSATURATED KETONES, CHALCONE AND TRANS-4-PHENYL-3-BUTEN-2-ONE, BY RAT LIVER MICROSOMES AND ESTROGENIC ACTIVITY OF THE METABOLITES
Drug Metab Dispos 2005 33: 1115-1123. Published online April 29, 2005; 10.1124/dmd.104.002634 [Abstract] [Full Text] [PDF]  

Mahesh N. Samtani, Matthias Lohle, Angela Grant, Peter W. Nathanielsz, and William J. Jusko
BETAMETHASONE PHARMACOKINETICS AFTER TWO PRODRUG FORMULATIONS IN SHEEP: IMPLICATIONS FOR ANTENATAL CORTICOSTEROID USE
Drug Metab Dispos 2005 33: 1124-1130. Published online April 28, 2005; 10.1124/dmd.105.004309 [Abstract] [Full Text] [PDF]  

Santosh Kumar, Dmitri R. Davydov, and James R. Halpert
ROLE OF CYTOCHROME B5 IN MODULATING PEROXIDE-SUPPORTED CYP3A4 ACTIVITY: EVIDENCE FOR A CONFORMATIONAL TRANSITION AND CYTOCHROME P450 HETEROGENEITY
Drug Metab Dispos 2005 33: 1131-1136. Published online May 3, 2005; 10.1124/dmd.105.004606 [Abstract] [Full Text] [PDF]  

Fanchon Bourasset, Katy Bernard, Carmen Muñoz, Patrick Genissel, and Jean-Michel Scherrmann
NEUROPHARMACOKINETICS OF A NEW {alpha}-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLE PROPIONIC ACID (AMPA) MODULATOR, S18986 [(S)-2,3-DIHYDRO-[3,4]CYCLOPENTANO-1,2,4-BENZOTHIADIAZINE-1,1-DIOXIDE], IN THE RAT
Drug Metab Dispos 2005 33: 1137-1143. Published online April 28, 2005; 10.1124/dmd.105.004424 [Abstract] [Full Text] [PDF]  

Undi Hoffler and Burhan I. Ghanayem
INCREASED BIOACCUMULATION OF URETHANE IN CYP2E1-/- VERSUS CYP2E1+/+ MICE
Drug Metab Dispos 2005 33: 1144-1150. Published online May 6, 2005; 10.1124/dmd.105.003806 [Abstract] [Full Text] [PDF]  

Naomi Morita, Hiroyuki Kusuhara, Yoshitane Nozaki, Hitoshi Endou, and Yuichi Sugiyama
FUNCTIONAL INVOLVEMENT OF RAT ORGANIC ANION TRANSPORTER 2 (SLC22A7) IN THE HEPATIC UPTAKE OF THE NONSTEROIDAL ANTI-INFLAMMATORY DRUG KETOPROFEN
Drug Metab Dispos 2005 33: 1151-1157. Published online May 17, 2005; 10.1124/dmd.104.001552 [Abstract] [Full Text] [PDF]  

Maciej J. Zamek-Gliszczynski, Keith A. Hoffmaster, Xianbin Tian, Rong Zhao, Joseph W. Polli, Joan E. Humphreys, Lindsey O. Webster, Arlene S. Bridges, J. Cory Kalvass, and Kim L. R. Brouwer
MULTIPLE MECHANISMS ARE INVOLVED IN THE BILIARY EXCRETION OF ACETAMINOPHEN SULFATE IN THE RAT: ROLE OF MRP2 AND BCRP1
Drug Metab Dispos 2005 33: 1158-1165. Published online April 28, 2005; 10.1124/dmd.104.002188 [Abstract] [Full Text] [PDF]  

Sharon E. Murphy, Vytautas Raulinaitis, and Kathryn M. Brown
NICOTINE 5'-OXIDATION AND METHYL OXIDATION BY P450 2A ENZYMES
Drug Metab Dispos 2005 33: 1166-1173. Published online April 28, 2005; 10.1124/dmd.105.004549 [Abstract] [Full Text] [PDF]  

Mark T. Poch, N. Shane Cutler, Garold S. Yost, and Ronald N. Hines
MOLECULAR MECHANISMS REGULATING HUMAN CYP4B1 LUNG-SELECTIVE EXPRESSION
Drug Metab Dispos 2005 33: 1174-1184. Published online May 17, 2005; 10.1124/dmd.105.004523 [Abstract] [Full Text] [PDF]  

Teruko Imai, Masumi Imoto, Hisae Sakamoto, and Mitsuru Hashimoto
IDENTIFICATION OF ESTERASES EXPRESSED IN CACO-2 CELLS AND EFFECTS OF THEIR HYDROLYZING ACTIVITY IN PREDICTING HUMAN INTESTINAL ABSORPTION
Drug Metab Dispos 2005 33: 1185-1190. Published online May 20, 2005; 10.1124/dmd.105.004226 [Abstract] [Full Text] [PDF]  

Kim A. Johnson and Chandra Prakash
METABOLISM, EXCRETION, AND PHARMACOKINETICS OF (3-{[4-TERT-BUTYL-BENZYL)-(PYRIDINE-3-SULFONYL)-AMINO]-METHYL}-PHENOXY)-ACETIC ACID, AN EP2 RECEPTOR-SELECTIVE PROSTAGLANDIN E2 AGONIST, IN MALE AND FEMALE SPRAGUE-DAWLEY RATS
Drug Metab Dispos 2005 33: 1191-1201. Published online May 10, 2005; 10.1124/dmd.105.004713 [Abstract] [Full Text] [PDF]  

Tatsuki Fukami, Miki Nakajima, Eriko Higashi, Hiroyuki Yamanaka, Haruko Sakai, Howard L. McLeod, and Tsuyoshi Yokoi
CHARACTERIZATION OF NOVEL CYP2A6 POLYMORPHIC ALLELES (CYP2A6*18 AND CYP2A6*19) THAT AFFECT ENZYMATIC ACTIVITY
Drug Metab Dispos 2005 33: 1202-1210. Published online May 17, 2005; 10.1124/dmd.105.004994 [Abstract] [Full Text] [PDF]  

Heng-Keang Lim, Nicholas Duczak, Jr., Linda Brougham, Michael Elliot, Krupa Patel, and Kelvin Chan
AUTOMATED SCREENING WITH CONFIRMATION OF MECHANISM-BASED INACTIVATION OF CYP3A4, CYP2C9, CYP2C19, CYP2D6, AND CYP1A2 IN POOLED HUMAN LIVER MICROSOMES
Drug Metab Dispos 2005 33: 1211-1219. Published online April 28, 2005; 10.1124/dmd.104.003475 [Abstract] [Full Text] [PDF] Data Supplement  

Xiao-fei Zhou, Xinning Yang, Qi Wang, Robert A. Coburn, and Marilyn E. Morris
EFFECTS OF DIHYDROPYRIDINES AND PYRIDINES ON MULTIDRUG RESISTANCE MEDIATED BY BREAST CANCER RESISTANCE PROTEIN: IN VITRO AND IN VIVO STUDIES
Drug Metab Dispos 2005 33: 1220-1228. Published online May 20, 2005; 10.1124/dmd.104.003558 [Abstract] [Full Text] [PDF]  

Anne-Laure Minn, Hélène Pelczar, Claire Denizot, Michel Martinet, Jean-Marie Heydel, Bernard Walther, Alain Minn, Hervé Goudonnet, and Yves Artur
CHARACTERIZATION OF MICROSOMAL CYTOCHROME P450-DEPENDENT MONOOXYGENASES IN THE RAT OLFACTORY MUCOSA
Drug Metab Dispos 2005 33: 1229-1237. Published online May 6, 2005; 10.1124/dmd.105.004085 [Abstract] [Full Text] [PDF]  

Priyamvada Chandra, Brendan M. Johnson, Peijin Zhang, Gary M. Pollack, and Kim L. R. Brouwer
MODULATION OF HEPATIC CANALICULAR OR BASOLATERAL TRANSPORT PROTEINS ALTERS HEPATOBILIARY DISPOSITION OF A MODEL ORGANIC ANION IN THE ISOLATED PERFUSED RAT LIVER
Drug Metab Dispos 2005 33: 1238-1243. Published online May 20, 2005; 10.1124/dmd.105.003665 [Abstract] [Full Text] [PDF]  

Jie Wan, Brian A. Carr, N. Shane Cutler, Diane L. Lanza, Ronald N. Hines, and Garold S. Yost
SP1 AND SP3 REGULATE BASAL TRANSCRIPTION OF THE HUMAN CYP2F1 GENE
Drug Metab Dispos 2005 33: 1244-1253. Published online April 28, 2005; 10.1124/dmd.105.004069 [Abstract] [Full Text] [PDF]  

Satoru Koyano, Yoshiro Saito, Hiromi Fukushima-Uesaka, Seiichi Ishida, Shogo Ozawa, Naoyuki Kamatani, Hironobu Minami, Atsushi Ohtsu, Tetsuya Hamaguchi, Kuniaki Shirao, Teruhiko Yoshida, Nagahiro Saijo, Hideto Jinno, and Jun-Ichi Sawada
FUNCTIONAL ANALYSIS OF SIX HUMAN ARYL HYDROCARBON RECEPTOR VARIANTS IN A JAPANESE POPULATION
Drug Metab Dispos 2005 33: 1254-1260. Published online April 28, 2005; 10.1124/dmd.105.004655 [Abstract] [Full Text] [PDF]  

Short Communications:

Alexander C Whitley, Douglas H. Sweet, and Thomas Walle
THE DIETARY POLYPHENOL ELLAGIC ACID IS A POTENT INHIBITOR OF hOAT1
Drug Metab Dispos 2005 33: 1097-1100. Published online May 3, 2005; 10.1124/dmd.105.004275 [Abstract] [Full Text] [PDF]  

To see an article, click its [Full Text] or [PDF] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.


Cover Caption:

Comparison of the structure and subcellular localization of NOSII and P450R. See the article by Riddick et al. on page 1083 of this issue.



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