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February 2006; 34 (2)   [Index by Author]  [Cover Caption]
       Articles
       Short Communications
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Table of Contents (PDF) | Editorial Board (PDF) | Front Matter (PDF) | Back Matter (PDF) |
To see an article, click its [Full Text] or [PDF] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.

Articles:

Robert J. Barbuch, Kristina Campanale, Chad E. Hadden, Milton Zmijewski, Ping Yi, Douglas D. O'Bannon, Jennifer L. Burkey, and Palaniappan Kulanthaivel
IN VIVO METABOLISM OF [14C]RUBOXISTAURIN IN DOGS, MICE, AND RATS FOLLOWING ORAL ADMINISTRATION AND THE STRUCTURE DETERMINATION OF ITS METABOLITES BY LIQUID CHROMATOGRAPHY/MASS SPECTROMETRY AND NMR SPECTROSCOPY
Drug Metab Dispos 2006 34: 213-224. Published online October 28, 2005; 10.1124/dmd.105.007401 [Abstract] [Full Text] [PDF]  

S. Sahasranaman, M. Issar, and G. Hochhaus
METABOLISM OF MOMETASONE FUROATE AND BIOLOGICAL ACTIVITY OF THE METABOLITES
Drug Metab Dispos 2006 34: 225-233. Published online October 26, 2005; 10.1124/dmd.105.005702 [Abstract] [Full Text] [PDF]  

Thomas K. H. Chang, Jie Chen, and Xiao Wei Teng
DISTINCT ROLE OF BILOBALIDE AND GINKGOLIDE A IN THE MODULATION OF RAT CYP2B1 AND CYP3A23 GENE EXPRESSION BY GINKGO BILOBA EXTRACT IN CULTURED HEPATOCYTES
Drug Metab Dispos 2006 34: 234-242. Published online October 28, 2005; 10.1124/dmd.105.005751 [Abstract] [Full Text] [PDF]  

Wenqing Gao, Zengru Wu, Casey E. Bohl, Jun Yang, Duane D. Miller, and James T. Dalton
CHARACTERIZATION OF THE IN VITRO METABOLISM OF SELECTIVE ANDROGEN RECEPTOR MODULATOR USING HUMAN, RAT, AND DOG LIVER ENZYME PREPARATIONS
Drug Metab Dispos 2006 34: 243-253. Published online November 4, 2005; 10.1124/dmd.105.007112 [Abstract] [Full Text] [PDF]  

Wenqing Gao, Jeffrey S. Johnston, Duane D. Miller, and James T. Dalton
INTERSPECIES DIFFERENCES IN PHARMACOKINETICS AND METABOLISM OF S-3-(4-ACETYLAMINO-PHENOXY)-2-HYDROXY-2-METHYL-N-(4-NITRO-3-TRIFLUOROMETHYLPHENYL)-PROPIONAMIDE: THE ROLE OF N-ACETYLTRANSFERASE
Drug Metab Dispos 2006 34: 254-260. Published online November 4, 2005; 10.1124/dmd.105.007120 [Abstract] [Full Text] [PDF]  

Ian S. Westley, Leonie R. Brogan, Raymond G. Morris, Allan M. Evans, and Benedetta C. Sallustio
ROLE OF MRP2 IN THE HEPATIC DISPOSITION OF MYCOPHENOLIC ACID AND ITS GLUCURONIDE METABOLITES: EFFECT OF CYCLOSPORINE
Drug Metab Dispos 2006 34: 261-266. Published online November 4, 2005; 10.1124/dmd.105.006122 [Abstract] [Full Text] [PDF]  

Donglu Zhang, Haiying Zhang, Nelly Aranibar, Ronald Hanson, Yande Huang, Peter T. Cheng, Shung Wu, Samuel Bonacorsi, Mingshe Zhu, Arun Swaminathan, and W. Griffith Humphreys
STRUCTURAL ELUCIDATION OF HUMAN OXIDATIVE METABOLITES OF MURAGLITAZAR: USE OF MICROBIAL BIOREACTORS IN THE BIOSYNTHESIS OF METABOLITE STANDARDS
Drug Metab Dispos 2006 34: 267-280. Published online November 9, 2005; 10.1124/dmd.105.007153 [Abstract] [Full Text] [PDF]  

Tooru Kamata, Munehiro Katagi, Hiroe T. Kamata, Akihiro Miki, Noriaki Shima, Kei Zaitsu, Mayumi Nishikawa, Einosuke Tanaka, Katsuya Honda, and Hitoshi Tsuchihashi
METABOLISM OF THE PSYCHOTOMIMETIC TRYPTAMINE DERIVATIVE 5-METHOXY-N,N-DIISOPROPYLTRYPTAMINE IN HUMANS: IDENTIFICATION AND QUANTIFICATION OF ITS URINARY METABOLITES
Drug Metab Dispos 2006 34: 281-287. Published online November 9, 2005; 10.1124/dmd.105.005835 [Abstract] [Full Text] [PDF] [Erratum]   

Kerry B. Goralski, Philip D. Acott, Albert D. Fraser, David Worth, and Christopher J. Sinal
BRAIN CYCLOSPORIN A LEVELS ARE DETERMINED BY ONTOGENIC REGULATION OF MDR1A EXPRESSION
Drug Metab Dispos 2006 34: 288-295. Published online November 22, 2005; 10.1124/dmd.105.007427 [Abstract] [Full Text] [PDF]  

Jen-Hung Yang, Te-Chun Hsia, Hsiu-Maan Kuo, Pei-Dawn Lee Chao, Chi-Chung Chou, Yau-Huei Wei, and Jing-Gung Chung
INHIBITION OF LUNG CANCER CELL GROWTH BY QUERCETIN GLUCURONIDES VIA G2/M ARREST AND INDUCTION OF APOPTOSIS
Drug Metab Dispos 2006 34: 296-304. Published online November 9, 2005; 10.1124/dmd.105.005280 [Abstract] [Full Text] [PDF]  

Vilasinee Hirunpanich, Jun Katagi, Benjabhorn Sethabouppha, and Hitoshi Sato
DEMONSTRATION OF DOCOSAHEXAENOIC ACID AS A BIOAVAILABILITY ENHANCER FOR CYP3A SUBSTRATES: IN VITRO AND IN VIVO EVIDENCE USING CYCLOSPORIN IN RATS
Drug Metab Dispos 2006 34: 305-310. Published online November 18, 2005; 10.1124/dmd.105.007088 [Abstract] [Full Text] [PDF]  

Sung Yeon Kim, Naomi Suzuki, Y. R. Santosh Laxmi, and Shinya Shibutani
INEFFICIENT REPAIR OF TAMOXIFEN-DNA ADDUCTS IN RATS AND MICE
Drug Metab Dispos 2006 34: 311-317. Published online November 18, 2005; 10.1124/dmd.105.007013 [Abstract] [Full Text] [PDF]  

Anubha Gupta, Pierre Chatelain, Roy Massingham, E. Niclas Jonsson, and Margareta Hammarlund-Udenaes
BRAIN DISTRIBUTION OF CETIRIZINE ENANTIOMERS: COMPARISON OF THREE DIFFERENT TISSUE-TO-PLASMA PARTITION COEFFICIENTS: Kp, Kp,u, AND Kp,uu
Drug Metab Dispos 2006 34: 318-323. Published online November 22, 2005; 10.1124/dmd.105.007211 [Abstract] [Full Text] [PDF]  

E. Row, S. A. Brown, A. V. Stachulski, and M. S. Lennard
DEVELOPMENT OF NOVEL FURANOCOUMARIN DIMERS AS POTENT AND SELECTIVE INHIBITORS OF CYP3A4
Drug Metab Dispos 2006 34: 324-330. Published online November 18, 2005; 10.1124/dmd.105.007294 [Abstract] [Full Text] [PDF]  

Hidetoshi Yamaya, Mayuko Saeki, Ken-ichiro Yoshida, Jiro Shibata, Shingo Yano, Yoshiaki Sato, Atsushi Takao, Takashi Shindo, Aman U. Buzdar, and Sekio Nagayama
DISTRIBUTION OF (7{alpha})-21-[4-[(DIETHYLAMINO) METHYL]-2-METHOXYPHENOXY]-7-METHYL-19-NORPREGNA-1,3,5(10)-TRIEN-3-OL-20-[14C]2-HYDROXY-1,2,3-PROPANETRICARBOXYLATE ([14C]TAS-108) AND ITS METABOLITES AFTER SINGLE ORAL ADMINISTRATION TO RATS BEARING 7,12-DIMETHYLBENZ({alpha})ANTHRACENE-INDUCED MAMMARY TUMOR
Drug Metab Dispos 2006 34: 331-338. Published online November 18, 2005; 10.1124/dmd.105.005504 [Abstract] [Full Text] [PDF]  

Short Communications:

Gwendolyn E. Kuehl, Jeannette Bigler, John D. Potter, and Johanna W. Lampe
GLUCURONIDATION OF THE ASPIRIN METABOLITE SALICYLIC ACID BY EXPRESSED UDP-GLUCURONOSYLTRANSFERASES AND HUMAN LIVER MICROSOMES
Drug Metab Dispos 2006 34: 199-202. Published online October 28, 2005; 10.1124/dmd.105.005652 [Abstract] [Full Text] [PDF]  

Johanna Weiss and Walter Emil Haefeli
EVALUATION OF INHIBITORY POTENCIES FOR COMPOUNDS INHIBITING P-GLYCOPROTEIN BUT WITHOUT MAXIMUM EFFECTS: F2 VALUES
Drug Metab Dispos 2006 34: 203-207. Published online November 4, 2005; 10.1124/dmd.105.007377 [Abstract] [Full Text] [PDF]  

Kazumi Sugihara, Yoshitaka Tayama, Kazuhiro Shimomiya, Daisuke Yoshimoto, Shigeru Ohta, and Shigeyuki Kitamura
ESTIMATION OF ALDEHYDE OXIDASE ACTIVITY IN VIVO FROM CONVERSION RATIO OF N1-METHYLNICOTINAMIDE TO PYRIDONES, AND INTRASPECIES VARIATION OF THE ENZYME ACTIVITY IN RATS
Drug Metab Dispos 2006 34: 208-212. Published online November 18, 2005; 10.1124/dmd.105.006544 [Abstract] [Full Text] [PDF]  

To see an article, click its [Full Text] or [PDF] link. To review many abstracts, check the boxes to the left of the titles you want, and click the 'Get All Checked Abstract(s)' button. To see one abstract at a time, click its [Abstract] link.


Cover Caption:

A schematic degradation pathway for conversion of MF into its degradation products D1, D2, and D3 on incubation of MF (C0 = 6.2µM) in plasma at 37°C for 72 h. See the article by Sahasranaman et al. on page 225 of this issue.



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